Synthesis and studying biological activity of new benzothiazole derivatives
نویسندگان
چکیده
A variety of novel tetrazole derivatives attached to the β-lactam ring was made utilizing heptanitrile in a reaction with generated azide-β-lactam derivatives, and these compounds were then studied using IR NMR spectroscopy. Biological testing showed that most final good antibacterial antifungal activity, particularly derivative (b3), which shown efficacy on par or even superior reference drugs Fluconazole Amoxicillin.
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ژورنال
عنوان ژورنال: Journal of Pharmaceutical Negative Results
سال: 2022
ISSN: ['0976-9234', '2229-7723']
DOI: https://doi.org/10.47750/pnr.2022.13.04.075